This paper explores the various aspects of workforce digitalization in Pakistan. Through an exploratory case study, it examines key trends of workforce digitalization, and the multifaceted impact of digitalization on the workforce in Pakistan, highlighting the opportunities, challenges, and economic benefits. Moreover, it analyzes the government policies and initiatives for the promotion of digitalization in Pakistan. Finally, it suggests a roadmap for workforce digitalization and economic transformation in Pakistan. Workforce digitalization and economic transformation entail a multifaceted approach to modernizing labor practices, leveraging digital technologies, and fostering economic growth. The digitalization of the workforce in Pakistan reflects the country’s evolving socio-economic landscape and technological advancements. However, workforce digitalization and economic transformation in Pakistan present significant opportunities and challenges. Embracing digitalization can enhance productivity, create new job opportunities, and drive economic growth. Further, modernizing government services through digitalization initiatives, including e-governance platforms for improved efficiency, transparency, and accountability fosters a more conducive environment and accelerates digital transformation across different sectors. However, addressing challenges related to digital literacy, cybersecurity, and access to digital infrastructure is essential to ensure that all segments of the population can benefit from the digital economy. As Pakistan seeks to strengthen its economy, digitalization is key to unlocking new opportunities, driving sustainable development, and becoming a digital nation in the future. Workforce digitalization and economic transformation in Pakistan require a comprehensive strategy that addresses digital skills development, infrastructure improvement, entrepreneurship support, government digitization, digital inclusion, cybersecurity, industry collaboration, and international partnerships. By prioritizing these areas, Pakistan can unlock its digital potential and drive sustainable economic growth in the digital age.