Pyridone Analogues Research Articles

Pyridone analogues of tetrahydroisoquinolines and protoberberines from mimosine and mimosinamine

Several pyrido[1,2-a]piperazines and their N-methyl derivatives have been prepared. These pyridine analogues of the 1,2,3,4-tetrahydroisoquinolines were formed by condensation of carbonyl compounds with mimosine and mimosinamine in the absence of an acid catalyst. A Mannich reaction converted one of these compounds, 1-(3,4-dimethoxybenzyl)-9-hydroxy-1,2,3,4-tetrahydro-8H-pyrido[1,2-a]- pyrazin-8-one, into a pyridone analogue of the tetrahydroprotoberberine caseadine.

ChemInform Abstract: POTENTIAL WOOL GROWTH INHIBITORS. 2(1H)‐PYRIDONE ANALOGS OF MIMOSINE

Chemischer InformationsdienstVolume 8, Issue 27 Natural Products ChemInform Abstract: POTENTIAL WOOL GROWTH INHIBITORS. 2(1H)-PYRIDONE ANALOGS OF MIMOSINE R. L. N. HARRIS, R. L. N. HARRISSearch for more papers by this authorT. TEITEI, T. TEITEISearch for more papers by this author R. L. N. HARRIS, R. L. N. HARRISSearch for more papers by this authorT. TEITEI, T. TEITEISearch for more papers by this author First published: July 5, 1977 https://doi.org/10.1002/chin.197727356AboutPDF ToolsRequest permissionExport citationAdd to favoritesTrack citation ShareShare Give accessShare full text accessShare full-text accessPlease review our Terms and Conditions of Use and check box below to share full-text version of article.I have read and accept the Wiley Online Library Terms and Conditions of UseShareable LinkUse the link below to share a full-text version of this article with your friends and colleagues. Learn more.Copy URL Share a linkShare onFacebookTwitterLinked InRedditWechat No abstract is available for this article. Volume8, Issue27July 5, 1977 RelatedInformation

Potential wool growth inhibitors. 2(1H)-Pyridone analogues of mimosine

The syntheses of DL-α-amino-β-(5-hydroxy-6-oxo-1,6-dihydropyridin-2- yl)propionic acid (3) and DL-α-amino-β-(1-hydroxy-2-oxo-1,2- dihydropyridin-4-yl)propionic acid (4), 2(1H)-pyridone isomers of the naturally occurring depilatory amino acid L-mimosine (1), are described.