Abstract
Aldimines (generated in situ from aldehydes and amines) undergo ready addition with ethyl diazoacetate in the presence of a catalytic amount of lithium perchlorate in acetonitrile to afford the corresponding cis-aziridine carboxylates in high yields with high diastereoselectivity. 10 mol% LiClO 4 in acetonitrile provides a convenient catalytic media to perform the reactions under mild and neutral conditions.
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