Abstract
A piperidinyl aziridine underwent alcoholic nucleophilic addition with alcohols to result in corresponding trans 3-amino-4-substituted piperidines. The addition reaction was catalyzed by BF 3·OEt 2 in excellent regio- and stereoselectivity. The application of this method was extended to the addition of thiols, acids and halogens with sustained regio- and stereoselectivity.
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