Abstract
AbstractWe have prepared a series of novel 2,3‐dihydro‐4‐pyridones containing boronate esters using the aza Diels–Alder reaction with Danishefsky's diene and imines derived from formylphenylboronic acids. This reaction can be carried out in moderate to high yields using Yb(OTf)3 as a Lewis acid catalyst. Two new boron compounds exhibited moderate antifungal activity (at 100 μg disk−1) using Amphotericin B as a control. © 2009 Wiley Periodicals, Inc. Heteroatom Chem 20:56–63, 2009; Published online in Wiley InterScience (www.interscience.wiley.com). DOI 10.1002/hc.20512
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