Abstract
In this article, an efficient, environmentally benign, one‐pot and simple synthesis of 2‐aryl/heteroarylbenzothiazoles by the reaction of 2‐aminothiophenol and aryl/heteroaryl aldehydes mediated by hypervalent iodine (III) reagents under solvent‐free condition at room temperature is demonstrated. All the reactions were carried out by grinding the reactants (2‐aminothiophenol and aryl/heteroaryl aldehydes) with hypervalent iodine (III) reagents in a mortar with pestle. Phenyliodine bistrifluoroacetate act as an efficient oxidizing reagent in comparison to iodobenzene diacetate in term of reaction time but yields are comparative. The advantages of this protocol are the one‐step procedure, mild reaction conditions, high yields of the products, and no side reactions.
Sign-in/Register to access full text options 
Talk to us
Join us for a 30 min session where you can share your feedback and ask us any queries you have
Schedule a callDisclaimer: All third-party content on this website/platform is and will remain the property of their respective owners and is provided on "as is" basis without any warranties, express or implied. Use of third-party content does not indicate any affiliation, sponsorship with or endorsement by them. Any references to third-party content is to identify the corresponding services and shall be considered fair use under The CopyrightLaw.
