Regioselective Suzuki coupling of benzofuran or benzothiophene boronic acids and dibromo substituted naphthalenes: synthesis of a potent inhibitor of plasminogen activator inhibitor-1

Zheng Wang,Hassan Elokdah,Geraldine Mcfarlane,Sherry Pan,Madelene Antane

doi:10.1016/j.tetlet.2006.03.090

Regioselective Suzuki coupling of benzofuran or benzothiophene boronic acids and dibromo substituted naphthalenes: synthesis of a potent inhibitor of plasminogen activator inhibitor-1

Zheng Wang, Hassan Elokdah + Show 3 more

https://doi.org/10.1016/j.tetlet.2006.03.090

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Journal: Tetrahedron Letters	Publication Date: Apr 11, 2006
Citations: 28

Affiliation: Princeton University

#Inhibitor Of Plasminogen Activator Inhibitor-1 #Regioselective Suzuki Coupling + Show 7 more

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Abstract

An efficient route to the biologically active naphthyl benzofuran derivative is described. The synthesis highlights a regioselective Suzuki coupling of a benzofuran and a dibromo substituted naphthalene. The scope of regioselective Suzuki coupling has been investigated.

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