Improved Procedure for the Solution Phase Preparation of 1,4-Benzodiazepine-2,5-dione Libraries via Armstrong's Convertible Isonitrile and the Ugi Reaction

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ADVERTISEMENT RETURN TO ISSUEPREVNoteNEXTImproved Procedure for the Solution Phase Preparation of 1,4-Benzodiazepine-2,5-dione Libraries via Armstrong's Convertible Isonitrile and the Ugi ReactionChristopher Hulme, John Peng, Sheng-Yuh Tang, Christopher J. Burns, Isabelle Morize, and Richard LabaudiniereView Author Information Lead Discovery Department, Rhône-Poulenc Rorer Central Research, 500 Arcola Road, Collegeville, Pennsylvania 19426-0995 Cite this: J. Org. Chem. 1998, 63, 22, 8021–8023Publication Date (Web):October 1, 1998Publication History Received3 April 1998Published online1 October 1998Published inissue 1 October 1998https://doi.org/10.1021/jo980622rCopyright © 1998 American Chemical SocietyRIGHTS & PERMISSIONSArticle Views1089Altmetric-Citations87LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InReddit Read OnlinePDF (76 KB) Get e-AlertsSUBJECTS:Aldehydes,Amines,Cyclization,Reagents,Solution phase Get e-Alerts