Abstract
Various N-substituted derivatives of glutamine, asparagine, glutaramic, succinamic and maleamic acids have been synthesized and tested in vitro against Plasmodium falciparum. From these compounds, only the glutamine derivatives ( 1–3) were found to have low activity. Kinetic evaluation of 1–3 revealed that these compounds also act as competitive inhibitors of γ-glutamyl transpeptidase (EC 2.3.2.2).
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