Abstract
AbstractAn approach to access bioactive thioamides was developed based on elemental‐sulfur‐promoted C(sp3)−H activation of methyl heteroarenes. This transformation could successfully furnish a series of heterocyclic thioamides with excellent yields and it could be conducted on gram scale with good reaction efficiency. Mechanistic studies showed that methyl heteroarenes reacted with dimethylamine released from DMF to form the desired thioamide through elemental‐sulfur‐promoted C−H activation.
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