Abstract
The efficiency of enantiomeric 1‐aminoindane and 1,2,3,4‐tetrahydro‐1‐naphthylamine as chiral auxiliaries in trans‐ß‐lactam formation via Staudinger cycloaddition is examined. Aromatic aldehydes possessing one, two, or three methoxyl groups are used as imine precursors, and the influence of their number and position on the reaction output is studied. A comparison with the results obtained from 1‐phenylethyl and 1‐(2‐naphthyl)ethylamine‐derived imines is performed.
Full Text 
Sign-in/Register to access full text options
Sign-in/Register to access full text options 
Published version (
Free)
Free) 
Talk to us
Join us for a 30 min session where you can share your feedback and ask us any queries you have
Schedule a call
