ChemInform Abstract: Synthesis of Aza and Carbocyclic β‐Carbolines for the Treatment of Alcohol Abuse. Regiospecific Solution to the Problem of 3,6‐Disubstituted β‐ and Aza‐β‐carboline Specificity.

Abstract

AbstractAn improved method is elaborated for the synthesis of azacarbolines (IV) and carbolines (VII) by a Buchwald—Hartwig amination followed by an intramolecular Heck‐type cyclization.