Abstract
An efficient method was developed for the synthesis of 1,3,4-trisubstituted pyrazolo[3,4-b]pyridines, 3H-pyrazolo[3,4-c]isoquinolines and 3H-pyrazolo[4,3-f][1,7]naphthyridines via intramolecular Heck reactions of imine derivatives of β-halovinyl/aryl aldehydes and 5-aminopyrazoles. This palladium acetate catalyzed reaction afforded good yields of these pyrazolo fused compounds under thermal conditions in the presence of xantphos as the ligand.
Talk to us
Join us for a 30 min session where you can share your feedback and ask us any queries you have
Schedule a callDisclaimer: All third-party content on this website/platform is and will remain the property of their respective owners and is provided on "as is" basis without any warranties, express or implied. Use of third-party content does not indicate any affiliation, sponsorship with or endorsement by them. Any references to third-party content is to identify the corresponding services and shall be considered fair use under The CopyrightLaw.
