ChemInform Abstract: One‐Pot Synthesis of Quinolin‐4(1H)‐one Derivatives by a Sequential Michael Addition—Elimination/Palladium‐Catalyzed Buchwald—Hartwig Amination Reaction.

Abstract

AbstractThe title synthesis uses chlorovinyl aromatic ketones [e.g. (I)] or bromovinyl aromatic ketones [e.g. (XIV)] and amines as starting material and the products can be obtained in good to excellent yields.