Abstract

We successfully prepared boroxazolidones by the reaction of diarylborinic acids substituted with electron-withdrawing groups and α-amino acids with various substituents under physiological conditions. β-Amino acids and the bioactive compound biocytin also formed related chelate compounds in good yields. Since the reaction proceeded smoothly under moderate conditions in the presence of other functional groups, it could be a powerful tool for the target identification of bioactive molecules.

Talk to us

Join us for a 30 min session where you can share your feedback and ask us any queries you have

Schedule a call

Disclaimer: All third-party content on this website/platform is and will remain the property of their respective owners and is provided on "as is" basis without any warranties, express or implied. Use of third-party content does not indicate any affiliation, sponsorship with or endorsement by them. Any references to third-party content is to identify the corresponding services and shall be considered fair use under The CopyrightLaw.