Approaching the Next Inflection in Peptide Therapeutics: Attaining Cell Permeability and Oral Bioavailability

Abstract

Cell Permeation and Oral Bioavailability. Peptide drug discovery has been a source of significant challenge, innovation, and achievement for several decades. This work highlights the breakthrough stage of drug discovery, providing a consolidated resource for drug hunters and academics pursuing peptide drug discovery and targeting challenging intracellular therapeutic targets. Specific articles describe hit finding, computational methods, binding affinity, and cellular permeability. Readers seeking to understand state-of-the-art peptide drug discovery and development, as well as those looking for areas of future growth, will find this volume useful.