Amidation and N-Boc Deprotection Process Improvement for the Preparation of 5-(1-Piperazinyl)benzofuran-2-carboxamide, a Key Intermediate of Vilazodone

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ADVERTISEMENT RETURN TO ISSUEPREVTechnical NoteAmidation and N-Boc Deprotection Process Improvement for the Preparation of 5-(1-Piperazinyl)benzofuran-2-carboxamide, a Key Intermediate of VilazodonePrasenjit Das, Bindu Srivastava, Sony Joseph, Hashim Nizar*, and Mohan PrasadView Author Information Chemical Research Division, Ranbaxy Research Laboratories, Gurgaon, Haryana 122001, India*E-mail: [email protected]; Telephone: 91-124-4011832.Cite this: Org. Process Res. Dev. 2014, 18, 5, 665–667Publication Date (Web):April 15, 2014Publication History Received28 February 2014Published online25 April 2014Published inissue 16 May 2014https://doi.org/10.1021/op500070tCopyright © 2014 American Chemical SocietyRIGHTS & PERMISSIONSArticle Views1629Altmetric-Citations7LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InReddit Read OnlinePDF (243 KB) Get e-AlertsSUBJECTS:Alcohols,Chemical reactions,High-performance liquid chromatography,Impurities,Organic reactions Get e-Alerts