A new method for the synthesis of n-(2-aminoethyl)azoles by alkylation of azoles with 2-alkyl-4,5-dihydrooxazoles

Abstract

Ring opening in 2-alkyl-4,5-dihydrooxazoles by the action of azoles gave intermediate N-(2-azolylethyl)alkanamides, whose hydrolysis afforded N-(2-aminoethyl)azoles.