Abstract
AbstractHerein, we present our findings on the synthesis of 3,4‐oxepino‐fused indoles by a two‐step reaction sequence involving an initial allylic substitution followed by Rh(III)‐catalyzed intramolecular [3+2] annulation via C−H activation starting from Morita‐Baylis‐Hillman (MBH) acetates of acetylenic aldehydes. The strategy is amenable to broad range of MBH acetates providing a facile access to 3,4‐oxepino‐fused indoles in good yield.
Sign-in/Register to access full text options 
Talk to us
Join us for a 30 min session where you can share your feedback and ask us any queries you have
Schedule a callDisclaimer: All third-party content on this website/platform is and will remain the property of their respective owners and is provided on "as is" basis without any warranties, express or implied. Use of third-party content does not indicate any affiliation, sponsorship with or endorsement by them. Any references to third-party content is to identify the corresponding services and shall be considered fair use under The CopyrightLaw.
