Abstract
As a joint meeting, the 26th Medicinal Chemistry Conference of GP2A and 32nd Journées Franco-Belges de Pharmacochimie took place between 13th and 15th June at Asnelles sur Mer (Normandie, France), providing a unique opportunity for a wide group of European medicinal chemists to engage. Topics included chemical tools for medicinal chemistry, protein-protein interactions, epigenetics, natural product-inspired molecules, computer-aided drug design, and new strategies for the design and development of drugs. s of invited lectures, proffered young researcher communications, flash communications and posters presented during the meeting are collected in this report.
Highlights
The Groupement des Pharmacochimistes de l’Arc Atlantique (GP2A) is a group of academic medicinal chemists working in universities and research institutes near the western coast of Europe
We demonstrated that the lead of the first generation of oligopyridines, named Pyridoclax, interacts directly with Mcl-1, releases its pro-apoptotic partners Bim and Bak and induces massive apoptosis at 25 μM concentration in combination with anti-Bcl-xL strategies in chemoresistant ovarian cancer cell lines
Synthesis and Biological Evaluation of Dibenzofuran Derivatives Inspired from Cercosporamide as K5.i7n.aDseesInighnib, iStoyrnsth(FesCis09a)nd Biological Evaluation of Dibenzofuran Derivatives Inspired from Cercosporamide
Summary
The Groupement des Pharmacochimistes de l’Arc Atlantique (GP2A) is a group of academic medicinal chemists working in universities and research institutes near the western coast of Europe (the “Atlantic Arc”) It was founded in 1992 with the aim of bringing together researchers in this area to exchange ideas and experiences. The “Journées Franco-Belges de Pharmacochimie” (JFB) is a widely recognized annual medicinal chemistry meeting This two-day symposium, whose first edition was held in 1986, aims to promote exchanges between medicinal chemists, mainly from France and Belgium. The major research topics that were presented included chemical tools for medicinal chemistry, protein-protein interactions, epigenetics, natural product-inspired molecules, computer-aided drug design, and new strategies for the design and development of drugs These presentations were in the forms of lectures by invited experts, proffered young researcher communications, posters with flash oral presentations and a large number of posters from young scientists, PhD students and postdoctoral researchers
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