Abstract
AbstractAn efficient base‐promoted approach for the synthesis of pyrido[1,2‐a]pyrimidinones from ynones and 2‐methylpyrimidin‐4‐ols have been developed via the C−N and C−C formation procedure. Diversely structural pyrido[1,2‐a]pyrimidinones were afforded in up to 95% yield for 29 examples. This reaction featured with advantages such as practical tandem procedure, wide functional group tolerance and metal‐free conditions, which has potential application in synthetic and medicinal chemistry.
Sign-in/Register to access full text options 
Talk to us
Join us for a 30 min session where you can share your feedback and ask us any queries you have
Schedule a callDisclaimer: All third-party content on this website/platform is and will remain the property of their respective owners and is provided on "as is" basis without any warranties, express or implied. Use of third-party content does not indicate any affiliation, sponsorship with or endorsement by them. Any references to third-party content is to identify the corresponding services and shall be considered fair use under The CopyrightLaw.
